Diacetate
Mostrando 1-12 de 172 artigos, teses e dissertações.
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1. Diacetate Naphthoquinone Derivatives Tethered to 1,2,3-Triazoles: Synthesis and Cytotoxicity Evaluation in Caco-2 Cells
Acetylated compounds prepared from naphthoquinones have been reported as antitumoral prodrugs. Exploring the synthetic versatility of the naphthoquinone and triazolic nuclei, herein we report a simple and efficient synthetic route to prepare a series of sixteen prodrugs prototype of 1,2,3-triazoles-naphthoquinodoic acetyl derivatives. The compounds 10a-10h a
Journal of the Brazilian Chemical Society. Publicado em: 2022
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2. TOWARDS BRAZIL AND CHINA CROSS-CULTURAL UNDERSTANDING AND TRANSNATIONAL COOPERATION
ABSTRACT Oxisols are important soils that have been converted from native vegetation to croplands, and can affect soil biological properties such as microbial biomass and enzyme activity. Thus, the aim of this study was to evaluate the changes on soil microbial biomass and enzyme activity when native vegetation (NV) was converted to cropland (CL), such as ma
Rev. Bras. Lit. Comp.. Publicado em: 2020-12
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3. Soil microbial biomass and enzyme activity in six Brazilian oxisols under cropland and native vegetation
ABSTRACT Oxisols are important soils that have been converted from native vegetation to croplands, and can affect soil biological properties such as microbial biomass and enzyme activity. Thus, the aim of this study was to evaluate the changes on soil microbial biomass and enzyme activity when native vegetation (NV) was converted to cropland (CL), such as ma
Bragantia. Publicado em: 2020-12
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4. Conservation system improves soil microbial quality and increases soybean yield in the Northeastern Cerrado
ABSTRACT The conservation tillage systems is based on the surface protection by crop residue and reduced soil disturbance. These two principles can favor the soil quality and promote sustainable agricultural systems. The study was developed with the objective of measure soil microbial biomass, soil basal respiration, enzymatic activity and soybean yield in c
Bragantia. Publicado em: 2020-12
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5. Evaluation of the physical and antifungal effects of chlorhexidine diacetate incorporated into polymethyl methacrylate
Abstract This study aimed to evaluate the physical properties and antifungal activities of polymethyl methacrylate (PMMA) acrylic resins after the incorporation of chlorhexidine diacetate salt (CDA). Methodology: First, acrylic resin specimens were fabricated with Vipi Cor® and DuraLay® resins with and without the incorporation of 0.5%, 1.0% or 2.0% CDA.
J. Appl. Oral Sci.. Publicado em: 10/01/2020
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6. Microbiological Indicators of Soil Quality Under Native Forests are Influenced by Topographic Factors
Abstract: Several microbiological indicators of soil quality present high sensitivity, but little is known about the influence of topographic factors on them. This work aimed to evaluate variability of biological indicators of soil quality across a hillslope under native forest and the influence of topographic factors on them. Four positions on a hillslope w
An. Acad. Bras. Ciênc.. Publicado em: 02/12/2019
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7. Is Increasing Doses of Imazapyr + Imazapic Detrimental to the Main Crop Rotation Alternatives to Flooded Rice?
RESUMO: A mistura formulada de imazapyr + imazapic é o principal herbicida usado para o controle de plantas daninhas em arroz no sistema Clearfield®. O uso contínuo de altas doses pode aumentar sua atividade residual no solo. O objetivo deste trabalho foi determinar a sensibilidade de culturas de cobertura e soja em rotação com arroz irrigado a diferent
Planta daninha. Publicado em: 02/12/2019
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8. In vitro genotoxicity of nitroimidazoles as a tool in the search of new trypanocidal agents
BACKGROUND Only benznidazole (Bnz) (1) and nifurtimox (Nfx) (2) are licensed for the treatment of Chagas disease although their safety and efficacy profile are far from ideal. Farmanguinhos from Fiocruz has developed seven nitroimidazole compounds (4-10) analogs of megazol (3). OBJECTIVES To evaluate whether the genotoxic effect of 3 was abolished in the
Mem. Inst. Oswaldo Cruz. Publicado em: 27/06/2019
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9. Chemo-Preventive Functions of Grape Seed Proanthocyanidin Extract against UV-Induced Intracellular Oxidative Stress and Tyrosinase Activity
Clinical studies have identified that an excessive exposure of UV light can cause oxidative stress (OS) and tyrosinase enzyme over-expression, which are associated with multiple diseases including atherosclerosis, cancers, diabetics, rheumatoid arthritis. In this study, we investigated the impact of grape seed proanthocyanidin (GSPE) on regulating OS and tyr
J. Braz. Chem. Soc.. Publicado em: 2018-08
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10. Rhodolirium andicola: a new renewable source of alkaloids with acetylcholinesterase inhibitory activity, a study from nature to molecular docking
ABSTRACT Acetylcholinesterase is an important target for control of neurodegenerative diseases causing cholinergic signaling deficit. Traditionally, galanthamine has been used as an Amaryllidaceae-derived acetylcholinesterase inhibitor, although new Amaryllidaceae plants could serve as source for better acetylcholinesterase inhibitors. Therefore, the objecti
Rev. bras. farmacogn.. Publicado em: 2018-01
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11. Insights into the intracellular mechanisms of citronellal in Candida albicans: implications for reactive oxygen species-mediated necrosis, mitochondrial dysfunction, and DNA damage
Abstract INTRODUCTION Citronellal (Cit) possesses antifungal activity and has possible implications for reactive oxygen species (ROS) generation in Candida albicans. In this study, the effects of Cit on ROS generation and the mechanisms by which Cit exerts anti-Candida effects were examined. METHODS A 2′,7′-dichlorodihydrofluorescein diacetate assay
Rev. Soc. Bras. Med. Trop.. Publicado em: 2017-08
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12. Reforestation of a Degraded Area with Eucalyptus and Sesbania: Microbial Activity and Chemical Soil Properties
ABSTRACT Mining activities generally affect soil quality, degrading it and creating the need for consistent environmental recovery efforts. This study evaluates the influence of monospecific and mixed stands of Sesbania virgata (S) and Eucalyptus camaldulensis (E) on the chemical properties and microbial activity of the soil in a degraded area by clay extrac
Rev. Bras. Ciênc. Solo. Publicado em: 10/07/2017